Butalbital



Butalbital
Systematic (IUPAC) name
5-(2-methylpropyl)-5-(2-propenyl)-
2,4,6(1
H,3H,5H)-pyrimidinetrione
Identifiers
CAS number 77-26-9
ATC code  ?
PubChem 2481
DrugBank APRD00266
Chemical data
O3 
Mol. mass 224.256
Pharmacokinetic data
Bioavailability well absorbed
Metabolism hepatic
Half life 35 hours
Excretion  ?
Therapeutic considerations
Pregnancy cat.

D(US)

Legal status

Schedule III(US)

Routes oral

Butalbital, 5-allyl-5-isobutylbarbituric acid, is a FDA approved for the treatment of tension headaches.

Combinations include:

  • butalbital and acetaminophen (trade names: Axocet, Bucet, Bupap, Cephadyn, Dolgic, Phrenilin, Phrenilin Forte, Sedapap)
  • butalbital, acetaminophen, and caffeine (trade names: Fioricet, Esgic, Esgic-Plus)
  • butalbital and aspirin (trade name: Axotal)
  • butalbital, aspirin, and caffeine (trade names Fiorinal, Fiormor, Fiortal, Fortabs, Laniroif)
  • butalbital, acetaminophen, caffeine, and codeine phosphate (Fioricet #3 with Codeine)
  • butalbital, Fiorinal #3 with Codeine)

 

Side effects

Side effects for any drug are difficult to predict, but commonly reported side effects for butalbital include:

  • Dizziness
  • Drowsiness
  • Intoxicated feeling
  • Light-headedness
  • Nausea
  • Sedation
  • Addiction
  • Severe impairment of judgement

There are other potential side effects; this list should not be considered all-inclusive.

Dangers and Risks

Butalbital is a physically and psychologically addictive barbiturate. Butalbital should not be mixed with alcohol due to increased risk of intoxication.

There are other potential risks; this list should not be considered all-inclusive.

Butalbital and Acetaminophen (Systemic). MedicinePlus Drug Information. Retrieved on December 31, 2006.

Controlled Substances in Schedule III. Drug Enforcement Administration (2007). Retrieved on 2007-01-13.

 
This article is licensed under the GNU Free Documentation License. It uses material from the Wikipedia article "Butalbital". A list of authors is available in Wikipedia.